Explain why benzene undergoes electrophilic substitution with concentrated nitric acid in the presence of concentrated sulfuric acid, rather than electrophilic addition, and identify the electrophile responsible for the reaction.

IB DP Chemistry Standard Level (2023 syllabus) — R3.3 Electron sharing reactions · Explain · 4 marks · View as Markdown

Written & reviewed by James Millett — Biology (Imperial College London), PGCE Science (University of Cambridge).

Benzene reacts with a mixture of concentrated nitric acid and concentrated sulfuric acid to form nitrobenzene. The reaction preserves the ring structure of benzene.

Model answer (4 marks)

Benzene has a delocalised π‑electron system that gives it aromatic stability. In the mixture of concentrated nitric and sulfuric acids, sulfuric acid protonates nitric acid to give the nitronium ion (NO₂⁺), the electrophile. The NO₂⁺ attacks the π‑electron cloud of benzene, forming a σ‑complex (arenium ion) that temporarily disrupts aromaticity. In the second step a proton is lost, restoring the delocalised system. Electrophilic addition would break the ring’s aromaticity completely and would require a highly unfavourable loss of the π‑electron system, so substitution is energetically preferred.

Examiner tips

  • State the electrophile (NO₂⁺) and how it is formed
  • Explain the role of benzene’s delocalised π system
  • Mention that addition would destroy aromaticity
  • Show that substitution restores aromaticity after proton loss

Common mistakes

  • Confusing the nitronium ion with a nitrous acid species
  • Claiming that addition is possible without noting loss of aromaticity
  • Omitting the role of proton loss to restore aromaticity

Mark scheme (4 marks)

  1. The electrophile is the nitronium ion (NO₂⁺), generated when sulfuric acid protonates nitric acid.
  2. Benzene has a delocalised pi electron system / ring of delocalised electrons above and below the plane that attracts electrophiles.
  3. Addition would disrupt / destroy the delocalised electron system / aromaticity, which is energetically unfavourable.
  4. Substitution allows the delocalised system / aromaticity to be restored / retained when the proton is lost in the second step, making it the preferred pathway.

Key terms in this question

electrophilic substitution

Related

More Electron sharing reactions questions

▶ Try answering this question with AI marking (free) →